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Search Results for " estradiol receptor "

Targets

14

Compounds

3

Natural Products

5

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T0168 Estradiol (cypionate) Depofemin,Estradiol cypionate Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Estradiol cypionate (Depofemin), the 17 β-cyclopentylpropinate ester of estradiol, inhibits ET-1 synthesis via estrogen receptor.
T2231 Estradiol dipropionate 17-Beta-Estradiol-3,17-Dipropionate Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Progesterone Receptor
Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol.
T0384 Estradiol benzoate Benzoestrofol,Benzhormovarine,Benovocylin Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Estradiol benzoate (Benzhormovarine) is the synthetic benzoate ester of estradiol, a steroid sex hormone vital to the maintenance of fertility and secondary sexual characteristics in females.
T1536 Promestriene 3-propyl ethyl,17B-methyl estradiol,Promestriano Estrogen/progestogen Receptor
Promestriene (3-propyl ethyl) (INN) is a synthetic estrogen and glucocorticoid used topically in a 1% cream formulation. It is described as a tropic agent and antiseborrheic.
T1579 Mestranol Devocin,Norquen,Menophase Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Mestranol (Devocin), a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
T2569 Chlorotrianisene tris(p-methoxyphenyl)chloroethylene,CTA,tri-p-anisylchloroethylene,TACE Estrogen Receptor/ERR , Estrogen/progestogen Receptor , COX
Chlorotrianisene (tri-p-anisylchloroethylene) is an orally bioavailable, highly lipophilic, synthetic triphenylethylene (TPE) derivative and selective estrogen receptor modulator (SERM), with predominantly estrogenic but...
T9604 Beta-Estradiol 17-hemisuccinate Estrogen Receptor/ERR
beta-Estradiol 17-hemisuccinate selectively stains estrogen receptor (ER)-rich cells.
T11399 Giredestrant GDC-9545 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Giredestrant (GDC-9545) potently competes with estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has anti-tumor activity. Giredestrant, a non-steroidal ER ligand,...
TP2010 Kisspeptin 10 (dog)
Endogenous ligand for the canine KISS1 receptor (Kisspeptin receptor or GPR54). Stimulates section of luteinizing hormone, follicle stimulating hormone and estradiol in vivo.
T36913 17-Epiestriol
17-Epiestriol is a metabolite of estrone .1It is formed from estroneviaa 16α-hydroxy estrone intermediate by reduction of the C-17 ketone. 17-Epiestriol binds to estrogen receptor α (ERα) and ERβ with relative binding af...
T70399 TTC-352
TTC-352 is an orally bioavailable selective human estrogen receptor alpha (ERalpha; ESR1; ERa) partial agonist (ShERPA), with potential antineoplastic activity. Upon administration, TTC-352 mimics the naturally-occurring...
T76222 HFSH-β-(33-53) (TFA)
hFSH-β-(33-53) TFA, a thiol-containing peptide representing the second follicle-stimulating hormone receptor (FSHR) binding domain, acts as an FSHR antagonist. It prevents FSH from binding to its receptor and partially p...
T60827 TPBM
TPBM is a potent inhibitor of estrogen receptor α (ERα). The IC 50 value of TPBM for 17β-estradiol (E2)-ERα is 9 μM. TPBM is not toxic to cells and reduces E2·ERα recruitment to an endogenous estrogen-responsive gene. TP...
T70309 Dicetrorelix pamoate
Dicetrorelix pamoate is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity. GnRH induces the production and release of luteinizing hormone (LH) and follicle stimulating hormone (FSH)...
Cat No. Product Name Synonyms Targets
T1048 Estradiol E2,17β-Estradiol,17β-Oestradiol,β-Estradiol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
Estradiol (E2) is a naturally occurring steroidal sex hormone that is essential for female fertility and maintenance of secondary sexual characteristics. Estradiol upregulates IL-6 expression through estrogen receptor be...
T1424 Ethynyl estradiol 17α-Ethynylestradiol,Ethinyl Estradiol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
Ethynyl estradiol is a semisynthetic alkylated ESTRADIOL with a 17-alpha-ethinyl substitution. It has high estrogenic potency when administered orally, and is often used as the estrogenic component in ORAL CONTRACEPTIVES...
T7299 β-Estradiol 17-acetate beta-estradiol 17-acetate,1,3,5(10)-Estratriene-3,17β-diol 17-acetate Estrogen Receptor/ERR , Others
β-Estradiol 17-acetate (1,3,5(10)-Estratriene-3,17β-diol 17-acetate) is a metabolite of estradiol.

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPJ-00762 ER alpha Protein, Human, Recombinant (His) Human E. coli
Estrogen Receptor is a major ligand-activated transcription factor belonging to the nuclear hormone receptor superfamily. Estrogen Receptor is composed of several domains important for hormone binding, DNA binding, and a...
TMPY-01660 SULT1E1 Protein, Human, Recombinant (His) Human E. coli
Estrogen sulfotransferase, also known as Sulfotransferase, estrogen-preferring, Sulfotransferase 1E1, SULT1E1 and ST1E1, is a cytoplasm enzyme that belongs to the sulfotransferase 1 family. Sulfotransferase enzymes catal...
TMPK-00716 RANKL/TNFSF11/CD254 Protein, Human, Recombinant (aa 63-244) Human HEK293 Cells
Receptor activator of nuclear factor x03BA;B (RANK) and its ligand (RANKL) have originally been described for their key roles in bone metabolism and the immune system. Subsequently, it has been shown that the RANKL-RANK ...
TMPK-00591 RANKL/TNFSF11/CD254 Protein, Mouse, Recombinant (aa 70-316, His) Mouse HEK293 Cells
Receptor activator of nuclear factor x03BA;B (RANK) and its ligand (RANKL) have originally been described for their key roles in bone metabolism and the immune system. Subsequently, it has been shown that the RANKL-RANK ...
TMPK-00717 RANKL/TNFSF11/CD254 Protein, Human, Recombinant (His & Flag) Human HEK293 Cells
Receptor activator of nuclear factor x03BA;B (RANK) and its ligand (RANKL) have originally been described for their key roles in bone metabolism and the immune system. Subsequently, it has been shown that the RANKL-RANK ...
TargetMol